Zoetis Rimadyl R 20 mg tablet, 20 adet. pakette

Zoetis Rimadyl R 20 mg tablet, 20 adet. pakette

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Zoetis Rimadyl R 20 mg, 20 tablet, köpeklerin tedavisine yönelik, ameliyat sonrası ağrı ve inflamatuar reaksiyonları hafifletmek için kullanılan, karaciğer aromalı tabletler formundaki steroidal olmayan antiinflamatuar bir ilaçtır. < p> farmakolojik özellikler< güçlü>< p> Rimadyl R'nin aktif maddesi olan Carprofen, antiinflamatuar, analjezik ve antipiretik etkilere sahiptir. Karprofen, araşidonik asit döngüsündeki siklooksijenazı inhibe eder. Bu durumda ilaç ağırlıklı olarak inflamasyonun gelişmesine yanıt olarak indüklenen COX2'yi etkiler. Bunun sonucunda iltihaba, şişmeye ve ağrıya neden olan inflamatuar prostaglandinlerin sentezi engellenir. Terapötik dozlarda karprofenin COX1 üzerinde çok daha zayıf bir etkisi vardır ve bu nedenle koruyucu prostaglandinlerin sentezi üzerinde neredeyse hiç etkisi yoktur. Bu nedenle, karprofen dokulardaki, özellikle de mide, bağırsak, böbrek ve trombositlerdeki normal fizyolojik süreçlere müdahale etmez.< p> Karprofen, gastrointestinal sistemden hızla emilir ve uygulamadan 1-3 saat sonra en yüksek plazma konsantrasyonlarına ulaşır ve biyoyararlanımı daha fazladır. %90'dan fazla. Köpeklerde yarı ömrü yaklaşık 8 saattir. Karprofen %99'dan fazla plazma proteinlerine bağlanır. İlaç karaciğerde metabolize edilir, esas olarak dışkıyla (yaklaşık %80) ve idrarla atılır.< p> saklama koşulları< güçlü>< p> İlacı üreticinin ağzı kapalı ambalajında, kuru bir yerde, ışıktan koruyarak saklayın. 2°C ile 25°C arasındaki sıcaklıklarda, çocukların erişemeyeceği yerlerde, gıda ve yemlerden uzak tutun.< p>NSAID (steroidal olmayan antiinflamatuar ilaç) grubundan karaciğer aromalı tabletler. Antiinflamatuar, analjezik ve antipiretik etkileri vardır. Kas-iskelet sisteminin akut ve kronik hastalıklarında, analjezide ve köpeklerde postoperatif ağrı ve şişliği azaltmak için anti-inflamatuar ajan olarak kullanılır.



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